{"id":963,"date":"2023-05-03T22:38:06","date_gmt":"2023-05-03T20:38:06","guid":{"rendered":"https:\/\/www.linkidoc.fr\/blog\/2023\/05\/03\/les-nanoparticules-de-bottlebrush-delivrent-des-medicaments-immunostimulants\/"},"modified":"2023-05-03T22:38:08","modified_gmt":"2023-05-03T20:38:08","slug":"les-nanoparticules-de-bottlebrush-delivrent-des-medicaments-immunostimulants","status":"publish","type":"post","link":"https:\/\/www.linkidoc.fr\/blog\/2023\/05\/03\/les-nanoparticules-de-bottlebrush-delivrent-des-medicaments-immunostimulants\/","title":{"rendered":"Les nanoparticules de Bottlebrush d\u00e9livrent des m\u00e9dicaments immunostimulants"},"content":{"rendered":"<div>\n<div class=\"wp-block-image\">\n<figure class=\"alignright size-full\"><noscript><img loading=\"lazy\" decoding=\"async\" width=\"466\" height=\"480\" src=\"https:\/\/www.linkidoc.fr\/blog\/wp-content\/uploads\/2023\/05\/Les-nanoparticules-de-Bottlebrush-delivrent-des-medicaments-immunostimulants.jpg\" alt=\"\" class=\"wp-image-1548346\"  \/><\/noscript><\/figure>\n<\/div>\n<p>Des chercheurs du MIT ont d\u00e9velopp\u00e9 un syst\u00e8me de nanoparticules con\u00e7u pour administrer des m\u00e9dicaments immunostimulants aux tumeurs.  Ces m\u00e9dicaments sont destin\u00e9s \u00e0 stimuler les cellules immunitaires \u00e0 proximit\u00e9 des tumeurs pour qu&rsquo;elles commencent \u00e0 d\u00e9truire les cellules tumorales, mais lorsqu&rsquo;ils sont administr\u00e9s par voie syst\u00e9mique, ils provoquent des effets secondaires limitant la dose inacceptables tels qu&rsquo;une inflammation syst\u00e9mique.  Ces particules ont la forme d&rsquo;un goupillon, le m\u00e9dicament inactif \u00e9tant conjugu\u00e9 au \u00ab squelette de la brosse \u00bb.  En ajustant la formulation des particules, les chercheurs peuvent affiner leur profil de lib\u00e9ration et ont pu cr\u00e9er des particules qui s&rsquo;accumuleront au niveau de la tumeur sans provoquer d&rsquo;effets secondaires ailleurs.<\/p>\n<p>Entra\u00eener notre syst\u00e8me immunitaire \u00e0 d\u00e9truire les tumeurs est une strat\u00e9gie th\u00e9rapeutique anticanc\u00e9reuse prometteuse, et pr\u00e9sente une certaine \u00e9l\u00e9gance par rapport aux chimioth\u00e9rapies traditionnelles.  Cependant, cette approche n&rsquo;est pas sans limites, avec des effets secondaires possibles tels que des niveaux \u00e9lev\u00e9s d&rsquo;inflammation syst\u00e9mique.  Il existe diff\u00e9rentes m\u00e9thodes d&rsquo;immunoth\u00e9rapie contre les tumeurs, et l&rsquo;une consiste \u00e0 administrer des m\u00e9dicaments \u00e0 petites mol\u00e9cules qui peuvent activer les cellules immunitaires et les stimuler \u00e0 commencer \u00e0 produire des cytokines qui provoqueront une r\u00e9ponse inflammatoire locale et aideront \u00e0 d\u00e9truire la tumeur.  <\/p>\n<p>C&rsquo;est du moins la th\u00e9orie.  En r\u00e9alit\u00e9, l&rsquo;administration de tels m\u00e9dicaments dans tout le corps risque de provoquer des niveaux \u00e9lev\u00e9s d&rsquo;inflammation syst\u00e9mique, incitant ces chercheurs \u00e0 d\u00e9velopper un syst\u00e8me de nanoparticules pour les d\u00e9livrer directement \u00e0 la tumeur.  Ces nanoparticules de goupillon comportent une colonne vert\u00e9brale centrale et des \u00ab poils \u00bb.  Les m\u00e9dicaments immunostimulants peuvent \u00eatre conjugu\u00e9s au squelette central sous une forme inactive, connue sous le nom de pro-m\u00e9dicament, en utilisant des lieurs chimiques qui peuvent \u00eatre cliv\u00e9s dans le corps, permettant aux chercheurs d&rsquo;affiner la lib\u00e9ration.<!-- ASYNC UAT M - 300x250(t,r) - --><\/p>\n<p><!-- END ASYNC UAT M - 300x250(t,r) --><\/p>\n<p>\u00ab\u00a0Notre biblioth\u00e8que de prom\u00e9dicaments de goupillon nous a permis de montrer un effet immunologique du contr\u00f4le de la cin\u00e9tique de l&rsquo;immunoth\u00e9rapie, nous permettant de stimuler les r\u00e9ponses immunitaires tout en minimisant les effets secondaires\u00a0\u00bb, a d\u00e9clar\u00e9 Sachin Bhagchandani, chercheur impliqu\u00e9 dans l&rsquo;\u00e9tude.  \u00ab\u00a0Ce type d&rsquo;approche ouvre des perspectives aux scientifiques qui souhaitent d\u00e9coupler la toxicit\u00e9 de certains agents d&rsquo;immunoth\u00e9rapie prometteurs.\u00a0\u00bb<\/p>\n<p>\u00c0 ce jour, les chercheurs ont test\u00e9 un panel de six formulations de nanoparticules qui ont toutes \u00e9t\u00e9 con\u00e7ues pour lib\u00e9rer une classe de m\u00e9dicaments immunostimulants appel\u00e9s imidazoquinol\u00e9ines (IMD) \u00e0 des taux l\u00e9g\u00e8rement diff\u00e9rents.  Dans un mod\u00e8le de tumeur de souris, les versions \u00e0 lib\u00e9ration moyenne et lente des particules n&rsquo;ont produit aucun effet secondaire, tout en ayant une efficacit\u00e9 significative dans la r\u00e9duction de la croissance tumorale, tandis que les particules \u00e0 lib\u00e9ration rapide ont provoqu\u00e9 une inflammation syst\u00e9mique.  <\/p>\n<p>\u00ab\u00a0Nos mol\u00e9cules ont pu r\u00e9duire ces effets en toute s\u00e9curit\u00e9 en contr\u00f4lant la quantit\u00e9 de m\u00e9dicament actif lib\u00e9r\u00e9e dans le sang\u00a0\u00bb, a d\u00e9clar\u00e9 Bhagchandani.  \u00ab\u00a0Si vous minimisez la lib\u00e9ration du compos\u00e9 actif l\u00e0-bas, vous pouvez obtenir des effets anti-tumoraux sur le site de la tumeur sans les effets secondaires syst\u00e9miques.\u00a0\u00bb<\/p>\n<p>\u00c9tudier dans la revue <em>Avanc\u00e9es scientifiques<\/em>: La cin\u00e9tique d&rsquo;ing\u00e9nierie de la lib\u00e9ration d&rsquo;agonistes TLR7\/8 \u00e0 partir de prom\u00e9dicaments brosse \u00e0 bouteille permet une stimulation immunitaire cibl\u00e9e sur la tumeur<\/p>\n<p>Via : MIT<\/p>\n<p><!--TrendMD v2.4.8--><\/div>\n","protected":false},"excerpt":{"rendered":"<p>Des chercheurs du MIT ont d\u00e9velopp\u00e9 un syst\u00e8me de nanoparticules con\u00e7u pour administrer des m\u00e9dicaments immunostimulants aux tumeurs. Ces m\u00e9dicaments<\/p>\n","protected":false},"author":1,"featured_media":964,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[1],"tags":[1294,1286,62,1295,12,318,1285],"class_list":["post-963","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-non-classe","tag-bottlebrush","tag-delivrent","tag-des","tag-immunostimulants","tag-les","tag-medicaments","tag-nanoparticules","generate-columns","tablet-grid-50","mobile-grid-100","grid-parent","grid-50"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.2 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Les nanoparticules de Bottlebrush d\u00e9livrent des m\u00e9dicaments immunostimulants - Blog Linkidoc : consultant e-sant\u00e9<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/www.linkidoc.fr\/blog\/2023\/05\/03\/les-nanoparticules-de-bottlebrush-delivrent-des-medicaments-immunostimulants\/\" \/>\n<meta property=\"og:locale\" content=\"fr_FR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Les nanoparticules de Bottlebrush d\u00e9livrent des m\u00e9dicaments immunostimulants - Blog Linkidoc : consultant e-sant\u00e9\" \/>\n<meta property=\"og:description\" content=\"Des chercheurs du MIT ont d\u00e9velopp\u00e9 un syst\u00e8me de nanoparticules con\u00e7u pour administrer des m\u00e9dicaments immunostimulants aux tumeurs. 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