{"id":1403,"date":"2023-08-23T01:42:35","date_gmt":"2023-08-22T23:42:35","guid":{"rendered":"https:\/\/www.linkidoc.fr\/blog\/2023\/08\/23\/systeme-dadministration-de-medicaments-pour-la-grossesse-extra-uterine\/"},"modified":"2023-08-23T01:42:36","modified_gmt":"2023-08-22T23:42:36","slug":"systeme-dadministration-de-medicaments-pour-la-grossesse-extra-uterine","status":"publish","type":"post","link":"https:\/\/www.linkidoc.fr\/blog\/2023\/08\/23\/systeme-dadministration-de-medicaments-pour-la-grossesse-extra-uterine\/","title":{"rendered":"Syst\u00e8me d&rsquo;administration de m\u00e9dicaments pour la grossesse extra-ut\u00e9rine"},"content":{"rendered":"<div>\n<figure class=\"wp-block-image size-full\"><noscript><img loading=\"lazy\" decoding=\"async\" width=\"770\" height=\"433\" src=\"https:\/\/www.linkidoc.fr\/blog\/wp-content\/uploads\/2023\/08\/Systeme-dadministration-de-medicaments-pour-la-grossesse-extra-uterine.jpg\" alt=\"\" class=\"wp-image-1551089\"  \/><\/noscript><\/figure>\n<p>Des chercheurs de l&rsquo;Universit\u00e9 d&rsquo;\u00c9tat de l&rsquo;Oregon ont d\u00e9velopp\u00e9 un syst\u00e8me d&rsquo;administration de m\u00e9dicaments destin\u00e9 \u00e0 traiter la grossesse extra-ut\u00e9rine.  Survenant souvent dans les trompes de Fallope, les grossesses extra-ut\u00e9rines ne sont pas viables et constituent la principale cause de d\u00e9c\u00e8s maternel au cours du premier trimestre.  Un m\u00e9dicament appel\u00e9 m\u00e9thotrexate peut \u00eatre administr\u00e9 pour mettre fin \u00e0 la grossesse, mais peut provoquer des effets secondaires graves aux concentrations requises.  Ces chercheurs ont con\u00e7u un v\u00e9hicule de d\u00e9livrance de nanoparticules pour le m\u00e9thotrexate, capable de lib\u00e9rer sa charge m\u00e9dicamenteuse \u00e0 proximit\u00e9 de l&rsquo;endroit o\u00f9 il est n\u00e9cessaire en r\u00e9pondant au glutathion, un tripeptide pr\u00e9sent en concentrations \u00e9lev\u00e9es dans les cellules placentaires.  Cette technologie signifie que des doses consid\u00e9rablement plus faibles de m\u00e9thotrexate peuvent \u00eatre utilis\u00e9es pour traiter une grossesse extra-ut\u00e9rine, r\u00e9duisant ainsi le risque d&rsquo;effets secondaires.<\/p>\n<p>Les chercheurs \u00e0 l&rsquo;origine de cette derni\u00e8re \u00e9tude rapportent qu&rsquo;entre 1 % et 2 % des grossesses dans le monde sont extra-ut\u00e9rines.  Ces grossesses s&rsquo;implantent presque toujours dans les trompes de Fallope, o\u00f9 elles peuvent provoquer de graves l\u00e9sions entra\u00eenant des h\u00e9morragies, et constituent la principale cause de d\u00e9c\u00e8s maternel au cours du premier trimestre.  Le m\u00e9thotrexate peut \u00eatre utilis\u00e9 pour traiter la grossesse extra-ut\u00e9rine et agit en inhibant la capacit\u00e9 des cellules embryonnaires \u00e0 se diviser.   <\/p>\n<p>Cependant, aux doses requises, le m\u00e9dicament peut provoquer des effets secondaires graves, notamment des l\u00e9sions r\u00e9nales, des naus\u00e9es, des vomissements, de la diarrh\u00e9e et des maladies pulmonaires.  De plus, le m\u00e9thotrexate ne parvient pas \u00e0 traiter avec succ\u00e8s la grossesse extra-ut\u00e9rine dans environ 10 % des cas, en grande partie \u00e0 cause du manque de m\u00e9dicament atteignant le site cible.  Ces probl\u00e8mes ont incit\u00e9 ces chercheurs \u00e0 d\u00e9velopper une m\u00e9thode plus cibl\u00e9e d\u2019administration du m\u00e9thotrexate, ce qui signifie des concentrations accrues dans le tissu cible et une exposition r\u00e9duite ailleurs.<!-- ASYNC UAT M - 300x250(t,r) - --><\/p>\n<p><!-- END ASYNC UAT M - 300x250(t,r) --><\/p>\n<p>\u00ab\u00a0D\u00e9velopper des m\u00e9dicaments capables de cibler des endroits sp\u00e9cifiques du corps reste l&rsquo;un des plus grands d\u00e9fis de la biom\u00e9decine\u00a0\u00bb, a d\u00e9clar\u00e9 Olena Taratula, chercheuse impliqu\u00e9e dans l&rsquo;\u00e9tude.  \u00ab La plupart des m\u00e9dicaments prescrits aujourd\u2019hui, y compris le m\u00e9thotrexate, n\u2019ont aucun moyen d\u2019agir uniquement sur des tissus ou des cellules sp\u00e9cifiques.  Lorsque les m\u00e9dicaments affectent les cellules saines, ils peuvent r\u00e9duire consid\u00e9rablement la qualit\u00e9 de vie d\u2019un patient \u2013 \u200b\u200bpensez aux effets graves de la chimioth\u00e9rapie comme les cheveux, la perte de la muqueuse intestinale, la formation d\u2019ulc\u00e8res, les naus\u00e9es, etc.<\/p>\n<p>Leur solution consiste \u00e0 utiliser des polym\u00e8res, qui sont des versions synth\u00e9tiques de v\u00e9sicules telles que les liposomes.  Les polym\u00e8res, cependant, sont fabriqu\u00e9s \u00e0 partir de polym\u00e8res plut\u00f4t que de lipides.  Cependant, ces nanoparticules int\u00e8grent un m\u00e9canisme intelligent pour garantir qu\u2019elles lib\u00e8rent leur charge m\u00e9dicamenteuse exactement l\u00e0 o\u00f9 elle est n\u00e9cessaire.  Ils r\u00e9agissent au glutathion, un tripeptide pr\u00e9sent en concentrations \u00e9lev\u00e9es dans les cellules placentaires, leur permettant de lib\u00e9rer le m\u00e9dicament \u00e0 proximit\u00e9 de la grossesse extra-ut\u00e9rine.  Nous esp\u00e9rons que cela conduira \u00e0 une administration tr\u00e8s cibl\u00e9e du m\u00e9dicament pour traiter la maladie tout en \u00e9tant doux pour le reste de la femme.    <\/p>\n<p>\u00c9tude dans un journal <em>Petit<\/em>: Polym\u00e8res de m\u00e9thotrexate sensibles au glutathion pour la gestion potentielle de la grossesse extra-ut\u00e9rine<\/p>\n<p>Via\u00a0: Universit\u00e9 d\u2019\u00c9tat de l\u2019Oregon<\/p>\n<p><!--TrendMD v2.4.8--><\/div>\n","protected":false},"excerpt":{"rendered":"<p>Des chercheurs de l&rsquo;Universit\u00e9 d&rsquo;\u00c9tat de l&rsquo;Oregon ont d\u00e9velopp\u00e9 un syst\u00e8me d&rsquo;administration de m\u00e9dicaments destin\u00e9 \u00e0 traiter la grossesse extra-ut\u00e9rine.<\/p>\n","protected":false},"author":1,"featured_media":1404,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[1],"tags":[1705,1707,1706,318,5,731],"class_list":["post-1403","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-non-classe","tag-dadministration","tag-extrauterine","tag-grossesse","tag-medicaments","tag-pour","tag-systeme","generate-columns","tablet-grid-50","mobile-grid-100","grid-parent","grid-50"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.2 - 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